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Global R&D Pipeline
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Global R&D Pipeline

Tau
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Total number of drugs
228
Phase II and later clinical stages
8.3%
Involving companies
271
Main therapeutic areas
Nervous System Diseases
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Molecule Info
R&D and Market Info
ADC Info
DrugDrug Name EnDrug TypeTreatment FieldMechanism of ActionOriginatorDeveloperIndicationHighest Development StageHighest Development Stage (China)Approved Countries/RegionsApproved TimeApproved Time (China)Special ReviewADC TypeADC LinkerADC PayloadADC DARDrug NameAntibody TypeADC Linking SiteOperation
Florquinitau F18Florquinitau F18Small molecule drug Diagnostic radiopharmaceuticalsNervous System Diseases Other DiseasesTAU modulators PET imagingMerck Sharp & Dohme Corp.Sinotau Pharmaceutical Group University of California Enigma Biomedical Group, Inc.NDA/BLAPhase 3---Fast Track(United States)----Florquinitau F18--
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Flortaucipir F-18Flortaucipir F-18Small molecule drug Diagnostic radiopharmaceuticalsNervous System Diseases Other DiseasesTAU modulatorsSiemens Healthineers AGAvid Radiopharmaceuticals, Inc. Eli Lilly Nederland BV PDRadiopharma, Inc.Approved-United States European Union Japan United Kingdom Iceland Liechtenstein Norway2020-05-28------Flortaucipir F-18--
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Alzheimer's disease vaccine(Axon Biochemicals BV)Alzheimer's disease vaccine(Axon Biochemicals BV)Therapeutic vaccine Genetically engineered subunit vaccine Conjugated vaccineNervous System Diseases Eye Diseases Other Diseases Endocrinology and Metabolic DiseaseTAU modulators ImmunostimulantsAxon Biochemicals BVAXON Neuroscience SEPhase 2---------Alzheimer's disease vaccine(Axon Biochemicals BV)--
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PBT-434PBT-434Small molecule drugNervous System Diseases Endocrinology and Metabolic Disease Other Diseases Congenital DisordersTAU inhibitors α-synuclein inhibitorsAlterity Therapeutics Ltd.Alterity Therapeutics Ltd.Phase 2----Fast Track(United States) Orphan Drug(European Union) Orphan Drug(United States)----PBT-434--
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MK-2214MK-2214Monoclonal antibodyNervous System Diseases Other DiseasesTAU inhibitorsMerck & Co., Inc.Merck Sharp & Dohme LLC Merck Sharp & Dohme Corp.Phase 2---------MK-2214--
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EtalanetugEtalanetugMonoclonal antibodyNervous System Diseases Other DiseasesTAU inhibitorsEisai Co., Ltd.Eisai, Inc. Eisai Co., Ltd.Phase 2/3----Fast Track(United States)----Etalanetug--
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[F-18]Flornaptitril[F-18]FlornaptitrilSmall molecule drug Diagnostic radiopharmaceuticalsNervous System Diseases Other DiseasesAPP inhibitors TAU modulators PET imagingCeremark Pharma LLC University of California, Los AngelesCeremark Pharma LLCPhase 3---------[F-18]Flornaptitril--
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ASN-90ASN-90Small molecule drugNervous System Diseases Eye Diseases Other Diseases Endocrinology and Metabolic DiseaseAPP inhibitors OGA inhibitors TAU inhibitorsAsceneuron SAFerrer Internacional SA Asceneuron SA Merck Serono SAPhase 2/3----Orphan Drug(United States)----ASN-90--
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Hydromethylthionine mesylateHydromethylthionine mesylateSmall molecule drugNervous System Diseases Endocrinology and Metabolic Disease Other DiseasesTAU inhibitorsTauRx Pharmaceuticals Ltd.TauRx Therapeutics Ltd. TauRx Pharmaceuticals Ltd.NDA/BLAPhase 3---Innovative Licensing and Access Pathway(United Kingdom) Orphan Drug(European Union) Orphan Drug(United States)----Hydromethylthionine mesylate--
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[18F]Florzolotau[18F]FlorzolotauSmall molecule drug Diagnostic radiopharmaceuticalsNervous System Diseases Endocrinology and Metabolic Disease Eye Diseases Other DiseasesTAU modulatorsAprinoia Therapeutics, Inc.Aprinoia Therapeutics, Inc. Celgene Corp.Phase 3Phase 3---Fast Track(United States)----[18F]Florzolotau--
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Total 228 data
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